Cardiovascular Peptides

Research peptides that influence cardiac function, vascular health, blood pressure regulation, and cardiovascular tissue repair.

Cardiovascular Peptides

This category covers peptides researched for their effects on the heart, blood vessels, and circulatory system. Cardiovascular peptides act through mechanisms including angiogenesis, cardiac tissue repair, blood pressure regulation, endothelial function, and metabolic modulation.

Complete Peptide Directory

Natriuretic & Blood Pressure Peptides

PeptideDescriptionPrimary Mechanism
ANPAtrial natriuretic peptide that regulates blood pressure and fluid balanceNPR-A receptor; natriuresis, vasodilation, RAAS suppression
BNPB-type natriuretic peptide; cardiac biomarker and vasodilatorNPR-A receptor; ventricular volume/pressure regulation; heart failure marker
Angiotensin 1-7Counter-regulatory peptide in the renin-angiotensin systemMas receptor; vasodilation, anti-fibrotic, anti-inflammatory
BradykininVasoactive peptide that mediates vasodilation and inflammationB2 receptor; NO release, vasodilation, vascular permeability

Vascular & Endothelial Peptides

PeptideDescriptionPrimary Mechanism
ApelinEndogenous peptide that regulates cardiovascular homeostasis and angiogenesisAPJ receptor; positive inotrope, vasodilator, angiogenic factor
AdrenomedullinVasodilatory peptide with cardioprotective and angiogenic propertiesCRLR/RAMP2 receptor; vasodilation, angiogenesis, organ protection
Urotensin-2Most potent vasoconstrictor peptide known; cardiovascular remodelingUT receptor; vasoconstriction, cardiac hypertrophy, vascular remodeling
VIPVasoactive intestinal peptide with vasodilatory and anti-inflammatory effectsVPAC receptors; coronary vasodilation, pulmonary hypertension research
VIP AnalogModified VIP with enhanced stability for cardiovascular applicationsVPAC receptor agonist with improved pharmacokinetics

Cardiac Repair & Protection

PeptideDescriptionPrimary Mechanism
CardiogenShort peptide bioregulator targeting cardiac tissue gene expressionMyocardial regeneration; age-related cardiac decline; Khavinson research
CAR PeptideCardiac-homing peptide that targets injured myocardiumSelective accumulation in ischemic cardiac tissue; drug delivery vehicle
UrocortinCRF-related peptide with potent cardioprotective effectsCRF2 receptor; inotropic support, cardioprotection during ischemia
C-PeptideProinsulin cleavage product with vascular and neuroprotective effectsGPR146 receptor; endothelial NO release; microvascular function

Common Research Themes

Natriuretic Peptide System: ANP and BNP are both endogenous regulators of blood pressure and fluid balance, but originate from different cardiac chambers (atria vs. ventricles) and serve as distinct clinical biomarkers.

RAAS Counter-Regulation: Angiotensin 1-7 acts as a natural counterbalance to the vasoconstrictive and pro-fibrotic effects of angiotensin II, representing a protective arm of the renin-angiotensin system.

Cardiac Regeneration: Cardiogen and CAR Peptide represent two distinct approaches — Cardiogen targets gene expression in cardiac tissue through bioregulatory mechanisms, while CAR Peptide serves as a homing peptide to deliver therapeutics to injured myocardium.

Angiogenesis: Apelin, Adrenomedullin, and VIP all promote new blood vessel formation through distinct pathways, making them relevant to ischemic tissue research and vascular repair.

Getting Started

If you are new to this category, we recommend starting with BPC-157 — the most widely studied peptide in this category with broad cytoprotective effects across cardiovascular and vascular systems. From there, explore related peptides through the See Also sections on each page to build a comprehensive understanding of the research landscape.

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